An tsara Corticosteroid domin Sake Saki Saki
Rayos ( prednisone ), wanda ake kira Lodotra a Turai, yana da tsarin jinkirtaccen jinkirin maganin ƙananan kashi. Rayos, wanda masana'antar Horizon Pharma ne, ya amince da shi a ranar 26 ga watan Yuli, 2012, don maganin cututtuka da kuma wasu alamomi.
Shaidar FDA ta dogara ne akan bayanan da aka kwatanta da kwayoyin pharmacokinetics (watau yadda ake amfani da miyagun ƙwayoyi, maye gurbinta, kawar da) daga Rayos don sake ba da labari, da kuma bayanai daga Cibiyar Circadian na Prednisone a RA (CAPRA-1 da 2 ) gwaji.
CAPRA-2 ya nuna cewa mutane masu fama da matsananciyar cututtuka wadanda suka kasance tare da Rayos sunyi tasiri sosai a cikin ka'idojin amsa ACR20 idan aka kwatanta da placebo, da mahimmancin cigaba a matakin karfin. CAPRA-1 yayi la'akari da cikakken lafiyar Rayos.
Shaidawa
Rayos ne corticosteroid tare da anti-inflammatory ko immunosuppressive effects amfani da su kula da wasu rashin lafiyar, dermatologic, endocrine, gastrointestinal, hematologic, neoplastic, tsarin juyayi, ophthalmologic, refin, numfashi, da kuma yanayi rheumatologic.
Game da yanayin rheumatologic, Rayos za'a iya amfani dashi don taimako na gajeren lokaci na wani ɓangare na ɓangaren aikin gobarar. Ana iya amfani da Rayos a wasu lokuta na spondylitis , dermatomyositis, polymyositis, rheumatica polymyalgia , cututtuka na psoriatic , reversing polychondritis, arthritis rheumatoid, Sjogren's syndrome , Lupus erythematosus tsarin , da kuma vascularitis .
Availability
Rayos yana samuwa a matsayin 1 mg., 2 MG., Da 5 MG. jinkirta-saki kwamfutar hannu.
Bayyanawa
Dole ne a yi la'akari da hankali tare da la'akari da rashin lafiya da cututtuka kuma ko marasa lafiya suna amfani da maganganun da ke cikin lokaci-lokaci. Hakan farko shine yawancin 5 mg. Rayos sau ɗaya a rana. Duk da haka, marasa lafiya a halin yanzu a kan sanarwa na iya buƙatar gyaran gyare-gyare don daidaitawa daidai lokacin canzawa zuwa Rayos.
Dole ne a dauki Rayos tare da abinci, kuma dole ne a ɗauki kwamfutar hannu duka. Don tabbatarwa, ya kamata a yi amfani da kashi mafi kyau mafi dacewa. Dole ne ya kamata a yi hankali.
Ayyukan Mugunta
Halin halayen halayen da ke haɗuwa da corticosteroid sun hada da riƙe da ruwa, tsayi a cikin karfin jini, sauyawa cikin haƙuri mai glucose, canjin yanayi, karbar kayan aiki, da kuma ci gaba da ci.
Akwai wasu halayen halayen da zasu iya yiwuwa wanda ake dangantawa da mafi yawan tsarin jiki. Cikakken bayani game da Rayos yana dauke da babban jerin. Hanyoyin halayyar ƙwayoyin cuta da ke hade da corticosteroids sun hada da osteonecrosis na femoral da kuma halayen hagu, osteoporosis , raunin tsoka, asarar muscle taro, maganin maganin ƙwaƙwalwar ƙwayar cuta, da kuma rushewa.
Contraindications
Rayos bazai yi amfani da marasa lafiya ba tare da sanannun hypersensitivity zuwa prednisone ko wasu sinadarai marasa aiki da suke cikin kwamfutar hannu.
Gargaɗi
- Magunguna, musamman ma wadanda aka bi da su don wani lokaci mai tsawo, ya kamata a kula da su ga hypothalamic-pituitary-suppression axis suppression, Cushing ta ciwo, da kuma hyperglycemia.
- Akwai matsala mai yawa zuwa sababbin kamuwa da cuta kuma ya kara yawan haɗari na ƙwaƙwalwa ko sake dawo da kamuwa da cuta a cikin marasa lafiya da aka bi da Rayos ko prednisone.
- Ya kamata a kula da matsa lamba na jini, da sodium da potassium.
- Akwai haɗarin ƙwayar cuta na ciwo na gastrointestinal, ciki har da perforation. Kwayar cututtuka na iya zama masked.
- Euphoria, rashin barci, sauyawa yanayi, canje-canje na mutum, da kuma matsanancin damuwa na iya faruwa. Cikin halin da ake ciki a halin kwakwalwa yana iya kara damuwa tare da amfani da prednisone.
- Ragewa a ƙasa mai yawa zai iya faruwa.
- Akwai wasu abubuwa masu illolin ciki har da cataracts, glaucoma, da kamuwa da cuta.
- Rayuwa ko ciwon maganin alurar rigakafi marasa rai ya kamata a baiwa marasa lafiya shan kashi na immunosuppressive na prednisone.
- Raunin tayi zai iya faruwa a farkon farkon shekaru uku.
Drug Interactions
Rayos na iya hulɗa da:
- Anticoagulants
- Magunguna masu ciwon sukari
- CYP3A4 inducers da masu hanawa
- Cyclosporine
- NSAIDs (kwayoyin anti-inflammatory marasa amfani)
Tabbatar cewa likitanka na san duk magunguna da kariyar da kake ɗauka a halin yanzu. Yana da mahimmanci don tantance yiwuwar hadarin gaske tare da yiwuwar samun magani tare da Rayos.
Menene Bambancin?
Ta yaya Rayos ya bambanta daga nan da nan ya saki lakabi? A gwajin gwaji, Rayos an gudanar da shi a karfe 10 na yamma tare da abinci. Yanayin da aka jinkirta daga Rayos ya ba da izinin maganin warkewa a cikin jini don faruwa lokacin da matakan cytokine suka karu a tsakiyar dare. Wannan tsari na aiki zai iya samar da mafi kyawun kulawa da kumburi a wasu marasa lafiya.
Sources
Rayos. Bayyana Bayani.
http://www.rayosrx.com/PI/RAYOS-Dawallafa-Information.pdf
Horizon Pharma ta sanar da FDA Approval of RAYOS® (prednisone) Rigar-Release Tablets ga Rheumatoid Arthritis da Multiple Ƙarin Indications. Horizon Pharma. Yuli 2012.
http://ir.horizon-pharma.com/releasedetail.cfm?ReleaseID=695983