Methimazole, Carbimazole da Propylthiouracil / PTU
Lokacin da glanden thyroid ya zama overactive - wani yanayin da aka sani da hyperthyroidism - gland shine samar da yawa thyroid hormone. Wannan, a biyun, na iya haifar da wasu cututtuka da dama, ciki har da bugun jini mai tsanani, hawan jini, damuwa, rashin barci, girgizawa, asarar nauyi, zazzabin rai, da kuma yawancin alamomi na maganin mikiya, da kuma ƙwayoyi masu kyau.
Babban mahimmanci ga hyperthyroidism shine jinsin magungunan magani wanda aka sani da kwayoyi antithyroid. Ana kuma kira magungunan Antithyroid a matsayin thioamides. Su ne kwayoyi da ake amfani dasu don maganin maganin thyroid - hyperthyroidism - ciki har da lokacin da thyroid ne mai rauni saboda sakamakon cutar Graves, mai guba mai guba mai guba, ko mai guba na nodules.
Antithyroid kwayoyi aiki ta hanyar toshe thyroid gland shine ya iya samar da biyu key thyroid hormones thyroxine (T4) da triiodothyronine (T3).
Babban magungunan antithyroid a Amurka ana samun methimazole da propylthiouracil (PTU). A waje Amurka, zaɓin su ne methimazole, carbimazole, da kuma PTU.
Methimazole
Dandalin antithyroid na methimazole inhibits thyroid daga amfani da aidin - yawanci daga abinci ko kari - don samar da hormone thyroid. Yana da magani ne wanda marasa lafiya ke dauka sau daya a rana.
Methimazole an kira shi da sunan thiamazole.
Ana amfani da wannan miyagun ƙwayoyi a duniya kuma ita ce magungunan antithyroid na farko da aka yi amfani da su a Amurka, inda akwai samuwa a ƙarƙashin sunan suna Tapazole.
Yawancin masana'antun suna bayar da nau'i na methimazole.
Carbimazole
Carbimazole magani ne wanda, lokacin da aka gudanar da shi, ya juya cikin miyagun ƙwayoyi methimazole a cikin jiki, saboda haka ya kasance daidai da aikin.
Mafi sanannun alama na carbimazole ne Neomercazole.
Neomercazole shine alamar kasuwanci ce mai suna carbimazole kuma an gina ta ta Amdipharm International (Birtaniya). An bada izini a miyagun ƙwayoyi a shekara ta 2004, kuma an sayar da shi a Birtaniya da Turai, amma ba a samuwa a cikin ko Amurka ba. Za ka iya ganin datasheet akan Neomercazole a nan. Ga wadansu albarkatun da yawa game da Neomercazole.
- Yanar Gizo na Drug Maker: Amdipharm
- Bayyana Bayani
Neomercazole Sinadaran : carbimazole Ph.Eur; lactose; masarar masara; sucrose; magnesium stearate; sucrose; talc; yankakken alkama; ferric oxide; propyl hydroxybenzoate; da gelatin.
Ƙarfiyar Rasu : 5 MG
Wasu Brands / Sunaye: Carbimazole yana samuwa a wasu ƙasashen Turai da Asiya karkashin sunayen sunaye: Atirozidina, Basolest, CG1, Carbimazole Spofa, Carbotiroid, Mertiran, Neo-Mercazole, Neo-Thyreostat, Neo-Tireol, da Tyrazol.
Propylthiouracil / PTU
Hanyar PTU ya rage jinkirin thyroid ta overproduction na thyroid hormone shi ne cewa shi inhibits thyroid gland shine daga amfani da aidin don samar da hormone thyroid. Har ila yau, inhibits da yin hira da hormone thyroid T4 cikin T3. PTU yana da ɗan gajeren lokaci, don haka marasa lafiya suna shan wannan magani ana yawan umurce su su dauki magani sau biyu zuwa sau uku a kowace rana don rage matakan hormone.
PTU yana da tasiri fiye da sauran kwayoyi da aka tattauna a nan, kuma ita ce likitan da aka fi so domin hyperthyroid din kawai a cikin wasu yanayi (a lokacin da aka fara ciki, tsananin hawan kaza da kuma a yayin da mai haƙuri yana fama da mummunan sakamako daga methimazole).
A Amurka, kawai PTU mai nau'i ne kawai akwai; babu sunayen alamun PTU da aka sayar a Amurka. Yawan kamfanoni suna samar da PTU.
Ƙarin Bayani
Ƙara koyo game da hyperthyroidism da jiyya, ciki har da magungunan antithyroid, a cikin wadannan albarkatu:
- Rashin Harkokin Hyperthyroidism / Abun lura da cututtuka
- Risks da cututtukan cututtuka da kuma Hyperthyroidism
- Tambayoyi da yawa akan cutar kutsawa da cututtuka
- 3 hanyoyin da za a bi da Hyperthyroidism
Sources:
Daily Med, Abincin Amurka da Drug Administration Database Database, Online
Gidajen FDA na Sadarwar Drug: Sabon Gargadi na Garkewa akan cutar hanta mai tsanani tare da propylthiouracil, Afrilu 21, 2010, Online
Ross, Douglas MD, "Bayanin lafiyar: Antithyroid kwayoyi," UpToDate . An sabunta ta karshe: Nuwamba 13, 2009