Methimazole / Tapazole don Cututtuka

Antithyroid Drugs amfani da su magance cututtuka da kuma Hyperthyroidism

Magunguna na Antithyroid - wanda ake kira thioamides - su ne magunguna waɗanda ke bi da maganin thyroid (hyperthyroidism) ta hanyar hana ƙwayar glandon thyroid don samar da hormone thyroid. Yayin da kake kula da maganin karoid wanda ya fi yawanci daga yanayin da aka sani da cutar Graves, yana da muhimmanci a rage jinkirin ƙwayar glandon maganin hormones na thyroid, musamman ma thyroxine (T4) da triiodothyronine (T3).

Magunguna na Antithyroid sunyi aiki ta hanyar sanya shi mafi wuyar jiki don amfani da amin, don haka ya hana jigilar hormones a cikin gland.

Antithyroid magani magani yana daya daga cikin jiyya na hyperthyroidism da cutar Graves. Sauran jiyya sun haɗa da maganin Idinin rediyo (RAI) da kuma cirewa duka ko ɓangare na glandon thyroid .

Akwai magungunan antithyroid guda biyu a halin yanzu a Amurka: propylthiouracil (PTU) da methimazole. A Amurka, ana daukar methimazole a matsayin likitan maganin antithyroid da aka fi so a mafi yawan yanayi.

Methimazole, wani lokaci ana kira thiamazole, inhibits thyroid daga amfani da aidin don samar da hormone thyroid. An dauki shi a matsayin kashi ɗaya a kowace rana.

Ana amfani da miyagun ƙwayoyi a duniya. A {asar Amirka, Tapazole ita ce kawai sunan sunan antityroid miyagun ƙwayoyi na methimazole. Akwai masu yawan masana'antun methimazole.

Tapazole

Tapazole ita ce sunan methimazole , da magungunan antithyroid da King Pharmaceuticals ya gina, Inc. FDA ta amince da Tapazole a shekarar 2000.

Tapazole Sinadaran : Methimazole USP; lactose monohydrate; magnesium stearate; sitaci (masara); pregelatinized sitaci; da talc.

Ƙarfi Akwai : 5 MG da 10 MG

Methimazole Generic (by Sandoz)

Sandoz, mamba ne na Kamfanin Kamfanonin Novartis, na sana'ar methimazole. FDA ta amince da shi a shekarar 2001.

Sandoz Methimazole Sinadaran: Methimazole USP; lactose monohydrate; magnesium stearate; sitaci (masara); da talc.

Ƙarfi Akwai: 5 MG da 10 MG

Generic Methimazole (by Cedar Pharmaceuticals LLC)

Cedar Pharmaceuticals LLC masana'antun sunadaran methimazole wanda United Research Laboratories ke rarraba. An samu amincewar FDA a shekarar 2005.

Cedar Pharmaceuticals Methimazole Sinadaran: Methimazole USP; Jirgin da aka yi wa manoma; magnesium stearate; dankalin turawa; da talc.

Ƙarfi Akwai: 5 MG, 10 MG, 15 MG, 20 MG

Generic Methimazole (by Activis Totowa)

Ayyukan Totowa LLC na kamfanin Activiti Totowa da aka samu a shekara ta 2007 ne aka samu amincewar FED.

Aikata Methimazole Sinadaran Methimazole USP; lactose monohydrate; magnesium stearate; sitaci pregelatinized; da talc.

Ƙarfin samuwa: 5 MG da 10 MG

Methimazole na Generic (by Caraco Pharmaceutical Laboratories)

Caraco Pharmaceutical Laboratories, Ltd. ta samar da tsarin methimazole wanda FDA ta yarda a shekarar 2007.

Caraco Methimazole Sinadaran: Methimazole USP; lactose monohydrate; Povidone; talc; croscarmellose; magnesium stearate; da masarar masara.

Ƙarfi Akwai: 5mg da 10mg

Methimazole Generic (ta hanyar Kamfanonin Kasuwanci)

Ta Kamfanin Kamfanonin Pharmaceutical ke samar da methimazole.

Sinadaran: Methimazole USP; lactose monohydrate; magnesium stearate; masarar masara; da talc.

Ƙarfi Akwai: 5 MG da 10 MG

Sources:

Daily Med, Cibiyar Abinci da Drug Administration Medication Database.

Kasuwancin Tsaro na Dandalin FDA: Sabon Gargajiya na Garkewa akan Raunin Laifin Rauni Tare da Propylthiouracil, Afrilu 21, 2010

Ross, Douglas MD, "Bayanin lafiyar: Antithyroid kwayoyi," UpToDate . An sabunta ta karshe: Nuwamba 13, 2009

Ƙarin bayani daga: Leslie Blumenberg